Description
| Description | CCG-63802 is a reversible small-molecule inhibitor of regulator of G protein signaling (RGS) proteins. CCG-63802 inhibits the interaction between RGS4 and Galpha with an IC50 value of 1.4 μM. |
| Targets&IC50 | RGS4:1.4 μM |
| In vitro | CCG-63802 inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with Gαo. |
| Molecular Weight |
450.51 |
| Formula | C26H18N4O2S |
| CAS No. | 620112-78-9 |
Storage
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Solubility Information
DMSO: 1.67 mg/mL (3.71 mM),
Sonication and heating are recommended.
