Description
Description | RTS-V5 is a dual inhibitor of HDAC/proteasome (IC50s: 6.9, 18, 15, 0.27, 0.53 μM for HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, respectively). |
Targets&IC50 | HDAC6:0.27 nM, HDAC8:0.53 nM, HDAC1:6.9 nM, HDAC3:15 nM, HDAC2:18 nM |
Molecular Weight |
525.6 |
Formula | C27H35N5O6 |
CAS No. | 2285346-31-6 |
Storage
Powder: -20°C for 3 years | In solvent: -80°C for 1 year